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Carfilzomib (CAS# 868540-17-4)

Ngwongwo kemịkalụ:

Usoro ihe omimi C40H57N5O7
Molar Mass 719.92
Njupụta 1.161
Ebe Na-agbaze 204-208 Celsius C
Ebe Boling 975.6± 65.0 °C(buru amụma)
Ebe mgbari 543.8 ℃
Solubility Soluble na DMSO (ruo 80 mg / ml) ma ọ bụ na ethanol (ruo 25 mg / ml).
Uzuoku nrịbama 0mmHg na 25ºC
Ọdịdị siri ike
Agba Ọcha
pKa 13.17± 0.46 (buru amụma)
Ọnọdụ Nchekwa -20°
Nkwụsi ike Stable maka afọ 1 site na ụbọchị ịzụrụ dị ka enyere ya. Enwere ike ịchekwa ngwọta na DMSO ma ọ bụ ethanol na -20 ° ruo otu izu.
Ntụgharị uche 1.551
Jiri Ndị na-egbochi Proteasomel, analogs nke epoxomicin

Nkọwa ngwaahịa

Mkpado ngwaahịa

Koodu HS 29337900

 

Okwu mmalite

Carfilzomib (PR-171) bụ onye na-egbochi proteasome na-enweghị ike ịgbanwe ya na IC50.


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